Compound Reference

MOTS-C

A mitochondrial-derived peptide studied for AMPK activation, insulin sensitization, and retrograde mitochondrial signaling in metabolic aging models.

Mitochondrial-derived peptide (MDP)C₁₀₁H₁₆₅N₃₁O₂₉Approx. 30 to 60 minutes (preclinical)
AMPK ActivationMetabolic RegulationInsulin SensitivityMitochondrial SignalingLongevity

Overview

MOTS-C (Mitochondrial ORF of the 12S rRNA type-C) is a 16-amino acid peptide encoded within the mitochondrial 12S rRNA, identified by Lee et al. in 2015. It is classified as a mitochondrial-derived peptide (MDP) and represents a class of bioactive peptides whose existence was only recognized in the 2010s. MOTS-C is produced in the mitochondria and translocates to the cytoplasm and nucleus under metabolic stress, activating AMPK and regulating glucose and lipid metabolism. Animal studies have documented anti-obesity effects, improved insulin sensitivity, and extended lifespan in mouse models. Its identification bridged mitochondrial biology and peptide hormone research.

Quick Reference

Sequence
CRQGSIVHIRGFR (16 amino acids)
Genetic origin
Encoded in mitochondrial 12S rRNA gene
Discovery
Lee et al., Cell Metabolism, 2015
Primary mechanism
AMPK activation via AICAR-related pathway, nuclear translocation
Purity standard
>=98% by HPLC
Mechanism

How It Works

MOTS-C activates AMPK through an AICAR-related metabolic pathway, promoting cellular metabolic flexibility including increased glucose uptake via GLUT4 translocation, enhanced mitochondrial fatty acid oxidation, and suppression of de novo lipogenesis. Under metabolic stress, it translocates to the nucleus where it regulates adaptive stress response gene networks. This retrograde mitochondrial-to-nuclear signaling mechanism is its defining biological feature.

Research Highlights

Key findings from the published preclinical literature.

1

AMPK Activation and Metabolic Flexibility

Lee et al. (Cell Metabolism, 2015) documented MOTS-C activation of AMPK via an AICAR-like mechanism in skeletal muscle cells, with downstream effects on glucose uptake, fatty acid oxidation, and metabolic gene expression.

2

Anti-Obesity Effects in Mouse Models

Mouse studies showed that MOTS-C administration reduced body fat accumulation in high-fat diet models and improved insulin sensitivity, with effects on adipose tissue metabolism and muscle glucose uptake documented in multiple independent studies.

3

Lifespan Extension in Animal Research

Preclinical studies in aging mouse cohorts have examined MOTS-C effects on healthspan and lifespan parameters, with some models documenting extended survival and improved metabolic markers in MOTS-C-treated aged animals.

4

Nuclear Translocation Under Stress

Research has documented MOTS-C translocation from mitochondria to the nucleus under conditions of metabolic stress, where it interacts with nuclear factor regulatory networks to activate adaptive stress response programs.

Frequently Asked Questions

Source This Compound

MOTS-C is available from Spartan Peptides at a minimum 98% HPLC-verified purity with batch-specific certificate of analysis. Domestic US supply, same-day dispatch before 2 PM EST. For in-vitro research use only.

All compounds are strictly for in-vitro research use only and not intended for human consumption.